SB202190
Contact us: [email protected]
SB202190 |
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MBS808173-5x5mg | MyBiosource | 5x5mg | EUR 745 |
SB202190 |
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SIH-473-25MG | Stressmarq | 25 mg | EUR 292 |
SB202190 |
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SIH-473-5MG | Stressmarq | 5 mg | EUR 76.8 |
SB202190 (FHPI) |
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A1632-100 | ApexBio | 100 mg | EUR 80 |
Description: MAPK Signaling|p38 |
SB202190 (FHPI) |
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A1632-5.1 | ApexBio | 10 mM (in 1mL DMSO) | EUR 44 |
Description: MAPK Signaling|p38 |
SB202190 (FHPI) |
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MBS575414-100mg | MyBiosource | 100mg | EUR 175 |
SB202190 (FHPI) |
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MBS575414-10mg | MyBiosource | 10mg | EUR 135 |
SB202190 (FHPI) |
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MBS575414-200mg | MyBiosource | 200mg | EUR 225 |
SB202190 (FHPI) |
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MBS575414-25mg | MyBiosource | 25mg | EUR 140 |
SB202190 (FHPI) |
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MBS575414-50mg | MyBiosource | 50mg | EUR 145 |
SB202190 (FHPI, 4-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-5-(4-pyridyl)-1H-imidazole) |
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MBS6023840-1mg | MyBiosource | 1(mg | EUR 345 |
SB202190 (FHPI, 4-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-5-(4-pyridyl)-1H-imidazole) |
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MBS6023840-25mg | MyBiosource | 25mg | EUR 400 |
SB202190 (FHPI, 4-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-5-(4-pyridyl)-1H-imidazole) |
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MBS6023840-5mg | MyBiosource | 5(mg | EUR 475 |
SB202190 (FHPI, 4-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-5-(4-pyridyl)-1H-imidazole) |
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MBS6023840-5x5mg | MyBiosource | 5x5mg | EUR 1990 |
SB-7720770 2HCl |
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562446 | MedKoo Biosciences | 5.0mg | EUR 400 |
SB4315242, Free Base [CAS# 301836-41-9] |
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S-7800 | LC LABORATORIES | 5 mg | EUR 48 |
SB-366791 |
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20-abx076632 | Abbexa |
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SB-366791 |
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abx076632-250l | Abbexa | 250 µl | EUR 131.25 |
SB-366791 |
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abx076632-500l | Abbexa | 500 µl | EUR 337.5 |
SB-202190 |
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abx076748-100l | Abbexa | 100 µl | EUR 93.75 |
SB-202190 |
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abx076748-1ml | Abbexa | 1 ml | Ask for price |
SB-202190 |
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abx076748-200l | Abbexa | 200 µl | EUR 187.5 |
SB-216763 |
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abx076766-100l | Abbexa | 100 µl | EUR 118.75 |
SB-216763 |
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abx076766-1ml | Abbexa | 1 ml | Ask for price |
SB-216763 |
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abx076766-200l | Abbexa | 200 µl | EUR 275 |
SB216763 |
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20-abx076766 | Abbexa |
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SB-431542 |
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abx076786-100l | Abbexa | 100 µl | EUR 143.75 |
SB-431542 |
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abx076786-1ml | Abbexa | 1 ml | Ask for price |
SB-431542 |
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abx076786-200l | Abbexa | 200 µl | EUR 312.5 |
SB431542 |
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20-abx076786 | Abbexa |
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SB-203580 |
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abx076800-100l | Abbexa | 100 µl | EUR 131.25 |
SB-203580 |
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abx076800-1ml | Abbexa | 1 ml | Ask for price |
SB-203580 |
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abx076800-200l | Abbexa | 200 µl | EUR 337.5 |
SB203580 |
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20-abx076800 | Abbexa |
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SB-715992 |
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2468-25 | Biovision | each | EUR 836.4 |
SB-715992 |
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2468-5 | Biovision | each | EUR 261.6 |
SB-431542 |
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1674-1 | Biovision | each | EUR 202.8 |
SB-431542 |
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1674-5 | Biovision | each | EUR 535.2 |
SB-525334 |
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2880-25 | Biovision | each | EUR 757.2 |
SB-525334 |
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2880-5 | Biovision | each | EUR 235.2 |
SB-225002 |
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abx282811-100g | Abbexa | 100 µg | Ask for price |
SB-225002 |
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abx282811-20g | Abbexa | 20 µg | EUR 131.25 |
SB-225002 |
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abx282811-50g | Abbexa | 50 µg | EUR 337.5 |
SB-525334 |
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abx282848-100g | Abbexa | 100 µg | Ask for price |
SB-525334 |
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abx282848-20g | Abbexa | 20 µg | EUR 131.25 |
SB-525334 |
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abx282848-50g | Abbexa | 50 µg | EUR 312.5 |
SB-705498 |
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abx283246-100g | Abbexa | 100 µg | Ask for price |
SB-705498 |
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abx283246-20g | Abbexa | 20 µg | EUR 143.75 |
SB-705498 |
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abx283246-50g | Abbexa | 50 µg | EUR 337.5 |
SB-742457 |
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9568-25 | Biovision | each | EUR 652.8 |
SB-742457 |
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9568-5 | Biovision | each | EUR 210 |
SB-590885 |
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406109 | MedKoo Biosciences | 50.0mg | EUR 450 |
SB505124 |
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406135 | MedKoo Biosciences | 5.0mg | EUR 90 |
SB239063 |
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406337 | MedKoo Biosciences | 5.0mg | EUR 310 |
SB-218078 |
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406348 | MedKoo Biosciences | 1.0mg | EUR 295 |
SB525334 |
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406415 | MedKoo Biosciences | 10.0mg | EUR 150 |
SB525334 |
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A5602-100 | ApexBio | 100 mg | EUR 384 |
Description: Tyrosine Kinase|ALK#TGF-β / Smad Signaling|TGF-βR1(ALK5) |
SB525334 |
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A5602-25 | ApexBio | 25 mg | EUR 120 |
Description: Tyrosine Kinase|ALK#TGF-β / Smad Signaling|TGF-βR1(ALK5) |
SB525334 |
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A5602-5 | ApexBio | 5 mg | EUR 40 |
Description: Tyrosine Kinase|ALK#TGF-β / Smad Signaling|TGF-βR1(ALK5) |
SB525334 |
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A5602-5.1 | ApexBio | 10 mM (in 1mL DMSO) | EUR 40 |
Description: Tyrosine Kinase|ALK#TGF-β / Smad Signaling|TGF-βR1(ALK5) |
SB525334 |
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A5602-S | ApexBio | Evaluation Sample | EUR 24 |
Description: Tyrosine Kinase|ALK#TGF-β / Smad Signaling|TGF-βR1(ALK5) |
SB705498 |
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A8519-10 | ApexBio | 10 mg | EUR 120 |
Description: Membrane Transporter/Ion Channel|TRPV1 |
SB705498 |
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A8519-5 | ApexBio | 5 mg | EUR 64 |
Description: Membrane Transporter/Ion Channel|TRPV1 |
SB705498 |
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A8519-5.1 | ApexBio | 10 mM (in 1mL DMSO) | EUR 70.4 |
Description: Membrane Transporter/Ion Channel|TRPV1 |
SB705498 |
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A8519-50 | ApexBio | 50 mg | EUR 520 |
Description: Membrane Transporter/Ion Channel|TRPV1 |
SB-216763 |
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401903 | MedKoo Biosciences | 10.0mg | EUR 150 |
SB-431542 |
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401910 | MedKoo Biosciences | 10.0mg | EUR 90 |
SB225002 |
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406514 | MedKoo Biosciences | 50.0mg | EUR 450 |
SB-408124 |
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E1KS1545 | EnoGene | 5mg | EUR 211.2 |
SB590885 |
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E1KS2220 | EnoGene | 10mg | EUR 362.4 |
SB743921 |
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B1590-10 | ApexBio | 10 mg | EUR 167.2 |
Description: Cell Cycle/Checkpoint|Ksp |
SB743921 |
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B1590-200 | ApexBio | 200 mg | EUR 1314.4 |
Description: Cell Cycle/Checkpoint|Ksp |
SB743921 |
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B1590-50 | ApexBio | 50 mg | EUR 516 |
Description: Cell Cycle/Checkpoint|Ksp |
SB239063 |
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B1699-25 | Biovision | each | EUR 652.8 |
SB239063 |
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B1699-5 | Biovision | each | EUR 210 |
SB-590885 |
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B1708-25 | Biovision | each | EUR 652.8 |
SB-590885 |
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B1708-5 | Biovision | each | EUR 210 |
SB-415286 |
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B1954-25 | Biovision | each | EUR 907.2 |
SB-415286 |
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B1954-5 | Biovision | each | EUR 274.8 |
SB273005 |
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B6003-25 | ApexBio | 25 mg | EUR 718.4 |
Description: Angiogenesis|Integrin |
SB273005 |
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B6003-5 | ApexBio | 5 mg | EUR 136 |
Description: Angiogenesis|Integrin |
SB505124 |
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B2289-10 | ApexBio | 10 mg | EUR 94.4 |
Description: ALK4/ALK5/ALK7 inhibitor |
SB505124 |
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B2289-50 | ApexBio | 50 mg | EUR 296.8 |
Description: ALK4/ALK5/ALK7 inhibitor |
SB-204490 |
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B2507-1 | Biovision | each | EUR 157.2 |
SB-204490 |
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B2507-5 | Biovision | each | EUR 418.8 |
SB-297006 |
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B2589-25 | Biovision | each | EUR 548.4 |
SB-297006 |
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B2589-5 | Biovision | each | EUR 183.6 |
SB-297006 |
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555605 | MedKoo Biosciences | 100.0mg | EUR 450 |
SB269652 |
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522353 | MedKoo Biosciences | 5.0mg | EUR 255 |
SB-366791 |
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522592 | MedKoo Biosciences | 50.0mg | EUR 250 |
SB-265610 |
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526278 | MedKoo Biosciences | 10.0mg | EUR 250 |
SB-222200 |
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526724 | MedKoo Biosciences | 50.0mg | EUR 450 |
SB-408124 |
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526763 | MedKoo Biosciences | 5.0mg | EUR 150 |
SB649868 |
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526934 | MedKoo Biosciences | 100.0mg | EUR 1550 |
SB-756050 |
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528518 | MedKoo Biosciences | 100.0mg | EUR 350 |
SB-242235 |
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510235 | MedKoo Biosciences | 10.0mg | EUR 285 |
SB-202190 |
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510242 | MedKoo Biosciences | 50.0mg | EUR 300 |
SB328437 |
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532664 | MedKoo Biosciences | 10.0mg | EUR 325 |
SB452533 |
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532670 | MedKoo Biosciences | 10.0mg | EUR 345 |
SB-204990 |
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551029 | MedKoo Biosciences | 1.0mg | EUR 225 |
SB203850 |
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555153 | MedKoo Biosciences | 10.0mg | EUR 265 |
SB-222200 |
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A3795-10 | ApexBio | 10 mg | EUR 96 |
Description: GPCR/G protein|NK3 Receptor |
SB-222200 |
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A3795-5.1 | ApexBio | 10 mM (in 1mL DMSO) | EUR 104 |
Description: GPCR/G protein|NK3 Receptor |
SB-222200 |
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A3795-50 | ApexBio | 50 mg | EUR 412.8 |
Description: GPCR/G protein|NK3 Receptor |
SB-674042 |
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A3800-10 | ApexBio | 10 mg | EUR 203.2 |
Description: GPCR/G protein|OX Receptor |
SB-674042 |
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A3800-25 | ApexBio | 25 mg | EUR 717.6 |
Description: SB-674042 is a specific, high-affinity OX1 selective antagonist. |
SB-674042 |
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A3800-5 | ApexBio | 5 mg | EUR 121.6 |
Description: GPCR/G protein|OX Receptor |
SB590885 |
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B1406-10 | ApexBio | 10 mg | EUR 96 |
Description: MAPK Signaling|Raf |
SB590885 |
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B1406-100 | ApexBio | 100 mg | EUR 624 |
Description: MAPK Signaling|Raf |
SB590885 |
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B1406-250 | ApexBio | 250 mg | EUR 1104 |
Description: MAPK Signaling|Raf |
SB590885 |
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B1406-5.1 | ApexBio | 10 mM (in 1mL DMSO) | EUR 120 |
Description: MAPK Signaling|Raf |
SB590885 |
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B1406-50 | ApexBio | 50 mg | EUR 384 |
Description: MAPK Signaling|Raf |
SB408124 |
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B2163-10 | ApexBio | 10 mg | EUR 68 |
Description: GPCR/G protein|OX Receptor |
SB408124 |
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B2163-100 | ApexBio | 100mg | EUR 432 |
Description: GPCR/G protein|OX Receptor |
SB408124 |
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B2163-25 | ApexBio | 25 mg | EUR 152 |
Description: GPCR/G protein|OX Receptor |
SB408124 |
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B2163-5 | ApexBio | 5 mg | EUR 40 |
Description: GPCR/G protein|OX Receptor |
SB408124 |
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B2163-50 | ApexBio | 50 mg | EUR 710.4 |
Description: SB408124 is a potent and novel nonpeptide antagonist of orexin-1 (OX(1)) receptor with Ki values of 27 nM and 57 nM in membrane formats and in whole cell, respectively. SB408124 was 50-fold selective over the human OX2 receptor [1]. |
SB271046 |
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B2255-10 | ApexBio | 10 mg | EUR 201.6 |
Description: SB-271046 is a selective and orally active 5-HT6 receptor antagonist.5-HT6 belongs to GPCR which stimulates adenylate cyclase via Gs, which cloned from rat striatum. |
SB271046 |
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B2255-50 | ApexBio | 50 mg | EUR 614.4 |
Description: SB-271046 is a selective and orally active 5-HT6 receptor antagonist.5-HT6 belongs to GPCR which stimulates adenylate cyclase via Gs, which cloned from rat striatum. |
SB271046 |
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B2255-S | ApexBio | Evaluation Sample | EUR 97.2 |
Description: SB-271046 is a selective and orally active 5-HT6 receptor antagonist.5-HT6 belongs to GPCR which stimulates adenylate cyclase via Gs, which cloned from rat striatum. |
SB742457 |
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B2256-25 | ApexBio | 25 mg | EUR 264 |
Description: GPCR/G protein|5-HT Receptor#Neuroscience|5-HT Receptor |
SB742457 |
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B2256-5 | ApexBio | 5 mg | EUR 84 |
Description: GPCR/G protein|5-HT Receptor#Neuroscience|5-HT Receptor |
SB742457 |
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B2256-5.1 | ApexBio | 10 mM (in 1mL DMSO) | EUR 125.6 |
Description: GPCR/G protein|5-HT Receptor#Neuroscience|5-HT Receptor |
SB-242235 |
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B2273-25 | Biovision | each | EUR 614.4 |
SB-242235 |
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B2273-5 | Biovision | each | EUR 210 |
SB-334867 |
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B1281-25 | ApexBio | 25 mg | EUR 324 |
Description: SB-334867 is a selective antagonist of orexin-1 receptor [1].Orexin-A and orexin-B are two peptides isolated from rat hypothalamus. They are involved in some physiological functions such as the control of feeding, energy metabolism and regulation of the sleep-wake cycle. |
SB-334867 |
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B1281-5.1 | ApexBio | 10 mM (in 1mL DMSO) | EUR 142.8 |
Description: SB-334867 is a selective antagonist of orexin-1 receptor [1].Orexin-A and orexin-B are two peptides isolated from rat hypothalamus. They are involved in some physiological functions such as the control of feeding, energy metabolism and regulation of the sleep-wake cycle. |
SB590885 |
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GW4213 | Glentham Life Sciences | 1mg | EUR 339.64 |
SB590885 |
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GW4213-1 | Glentham Life Sciences | 1 | EUR 171.5 |
SB590885 |
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GW4213-10 | Glentham Life Sciences | 10 | EUR 318.6 |
SB590885 |
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GW4213-5 | Glentham Life Sciences | 5 | EUR 254 |
SB-242235 |
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GW7595 | Glentham Life Sciences | 1mg | EUR 1151.82 |
SB-242235 |
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GW7595-1 | Glentham Life Sciences | 1 | EUR 351.7 |
SB-242235 |
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GW7595-10 | Glentham Life Sciences | 10 | EUR 1035.7 |
SB-242235 |
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GW7595-5 | Glentham Life Sciences | 5 | EUR 673.7 |
SB-224289 |
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HY-101105 | MedChemExpress | Get quote | Ask for price |
Description: SB-224289 is a selective 5-HT1B receptor antagonist, with anxiolytic effect[1]. |
SB-568849 |
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HY-100308 | MedChemExpress | 10mg | EUR 3370.8 |
Description: SB-568849 is a melanin-concentrating hormone receptor 1 (MCH R1) antagonist with a pKi of 7.7. |
SB-366791 |
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GL6242 | Glentham Life Sciences | 5mg | EUR 273.72 |
SB-366791 |
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GL6242-25 | Glentham Life Sciences | 25 | EUR 298.9 |
SB-366791 |
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GL6242-25MG | Glentham Life Sciences | 25 mg | EUR 385.2 |
SB-366791 |
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GL6242-5 | Glentham Life Sciences | 5 | EUR 104.3 |
SB-366791 |
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GL6242-5MG | Glentham Life Sciences | 5 mg | EUR 157.2 |
SB-525334 |
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GL1664 | Glentham Life Sciences | 5mg | EUR 97.14 |
SB-334867 |
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HY-10895 | MedChemExpress | 50mg | EUR 557.37 |
Description: SB-334867 (SB 334867A) is an excellent,selective and blood–brain barrier permeable orexin-1 (OX1) receptor antagonist, shows selectivity over OX2 (pKb=7.4), 100-fold over 5-HT2B, 5-HT2C with pKi values of 5.4 and 5.3, respectively[1]. SB-334867 reduces ethanol consumption and inhibits the acquisition of morphine-induced sensitization to locomotor activity in vivo[2][3]. |
SB-674042 |
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HY-10898 | MedChemExpress | 10mM/1mL | EUR 141.78 |
Description: SB-674042 is a potent and selective non-peptide orexin OX1 receptor antagonist (Kd=5.03 nM), exhibits 100-fold selectivity for OX1 over OX2 receptors with IC50 values of 3.76 nM and 531 nM, respectively[1][4]. |
SB-590885 |
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HY-10966 | MedChemExpress | 10mM/1mL | EUR 671.01 |
Description: SB-590885 is a potent B-Raf inhibitor with Ki of 0.16 nM, and has 11-fold greater selectivity for B-Raf over c-Raf, without inhibition to other human kinases. |
SB-734117 |
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HY-114005 | MedChemExpress | 1mg | EUR 342 |
Description: SB-734117 is a human cytomegalovirus (HCMV) replication inhibitor that prevents CREB and histone H3 post-translational modifications[1]. |
SB-206606 |
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HY-117239 | MedChemExpress | Get quote | Ask for price |
Description: SB-206606, a stereoisomer of BRL 37344, is a potentially specific, beta 3-adrenergic receptor (β3-AR) ligand. The affinity of [3H]SB 206606 is 76 times higher for the β3-AR than for the beta 1/beta 2-adrenergic receptors[1]. |
SB-429201 |
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HY-119017 | MedChemExpress | 10 mg | EUR 2326.88 |
Description: SB-429201 is a potent and selective HDAC1 (IC50~1.5 μM). SB-429201 displays at least a 20-fold preference for HDAC1 inhibition over HDAC3 and HDAC8[1][2]. |
SB357134 |
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HY-119061 | MedChemExpress | Get quote | Ask for price |
Description: SB-357134 is a potent, selective, brain penetrant, and orally active 5-HT6 receptor antagonist. SB-357134 enhances memory and learning and increases seizure threshold in rats[1]. |
SB203580 |
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inh-sb20-5 | InvivoGen FR | 5 x 5 mg | EUR 136.5 |
SB-423562 |
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HY-15105 | MedChemExpress | 10mg | EUR 1049.8 |
Description: SB-423562 is a short-acting calcium-sensing receptor (CaR) antagonist. SB-423562 has the potential for osteoporosis research. |
SB-423557 |
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HY-15106 | MedChemExpress | Get quote | Ask for price |
Description: SB-423557 is an orally active calcium-sensing receptor (CaR) antagonist (IC50=520 nM), precursor of SB-423562 (IC50=73 nM). SB-423557 is well tolerated in human and increases plasma concentrations of exogenous parathyroid hormone (PTH) and stimulates bone formation[1]. |
SB-505124 |
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HY-13521 | MedChemExpress | 50mg | EUR 514.08 |
Description: SB-505124 is a selective inhibitor of TGF-β Receptor type I receptors (ALK4, ALK5, ALK7), with IC50s of 129 nM and 47 nM for ALK4, ALK5, respectively, but it does not inhibit ALK1, 2, 3, or 6. |
SB-222200 |
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HY-15722 | MedChemExpress | 10mg | EUR 799.8 |
Description: SB-222200 is a potent, selective, orally active and blood-brain barrier (BBB) penetrant NK-3 receptor antagonist. SB-222200 is developed for central nervous system (CNS) disorders[1]. |
SB-265610 |
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HY-50688 | MedChemExpress | 10mM/1mL | EUR 854.99 |
Description: SB-265610 is a selective, competitive, nonpeptide and allosteric CXCR2 antagonist. SB-265610 blocks rat cytokine-induced neutrophil chemoattractant-1 (CINC-1)-induced calcium mobilization and neutrophil chemotaxis with IC50s of 3.7 nM and 70 nM, respectively[1][2]. |
SB-408124 |
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HY-70068 | MedChemExpress | 10mM/1mL | EUR 73.59 |
Description: SB-408124 is a non-peptide OX1 receptor antagonist with Kis of 57 nM and 27 nM in whole cell and membrane, respectively. SB-408124 exhibits 50-fold selectivity over OX2 receptor[1]. |
SB225002 |
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HY-16711 | MedChemExpress | 100mg | EUR 345.24 |
Description: SB225002, a potent, selective and non-peptide CXCR2 antagonist, inhibits 125I-IL-8 binding to CXCR2 with an IC50 of 22 nM. |
SB-332235 |
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HY-16981 | MedChemExpress | 10 mg | EUR 651.53 |
Description: SB-332235 is a potent, orally active nonpeptide CXCR2 antagonist, with an IC50 of 7.7 nM. SB-332235 displays 285-fold selectivity for CXCR2 over CXCR1. SB-332235 inhibits acute and chronic models of arthritis in the rabbit. SB-332235 inhibits viability of AML cells[1][2]. |
SB-215505 |
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HY-18596 | MedChemExpress | Get quote | Ask for price |
Description: SB-215505 is a potent and subtype-selective 5-HT2B receptor antagonist with pKi values of 8.3, 6.77, 7.66 for 5-HT2B, 5-HT2A, 5-HT2C, respectively[1]. SB-215505 increases wakefulness and motor activity in rats[2]. |
SB-612111 |
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HY-18618 | MedChemExpress | Get quote | Ask for price |
Description: SB-612111 is a novel and potent opiate receptor-like orphan receptor (ORL-1) antagonist with a high affinity for hORL-1 (Ki=0.33 nM). SB-612111 exhibits selectivity for μ-, κ- and δ-receptors with Ki values of 57.6 nM, 160.5 nM and 2109 nM, respecticely. SB-612111 effectively antagonizes the pronociceptive action of Nociceptin (HY-P0183) in an acute pain model[1]. |
SB-209670 |
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HY-19210 | MedChemExpress | 1mg | EUR 617.98 |
Description: SB-209670 is an extremely potent and highly specific non-peptide, subnanomolar endothelin (ET) receptor antagonist. SB 209670 selectively inhibits binding of 125I-labeled ET-1 to cloned human ET receptor subtypes ETA and ETB (Ki=0.2 and 18 nM, respectively). SB 209670 produces a dose-dependent reduction in blood pressure in hypertensive rats, protects from ischemia-induced neuronal degeneration in a gerbil stroke model, and attenuates neointima formation following rat carotid artery balloon angioplasty[1]. |
SB-267268 |
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HY-19306 | MedChemExpress | 1 mg | EUR 2759.78 |
Description: SB-267268 is a selective and nonpeptidic alpha(v)beta3 (αvβ3) and alpha(v)beta5 (αvβ5) integrins antagonist, with Kis of 0.9, 0.5 and 0.7 nM for human αvβ3, monkey αvβ3 and human αvβ5, respectively. SB-267268 inhibits human and mouse αvβ3 with IC50s of 0.68 and 0.29 nM, respectively. SB-267268 reduces angiogenesis and VEGF expression[1]. |
SB-273005 |
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HY-19307 | MedChemExpress | 1 mg | EUR 811.7 |
Description: SB-273005 is a potent nonpeptide and orally active integrin antagonist with Kis of 1.2 nM and 0.3 nM for αvβ3 receptor and αvβ5 receptor, respectively[1]. |
SB-435495 |
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HY-19415 | MedChemExpress | 10 mg | EUR 974.04 |
Description: SB-435495 is a potent, selective, reversible, non-covalent and orally active Lp-PLA2 inhibitor with an IC50 of 0.06 nM[1][3]. |
SB-649701 |
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HY-153669 | MedChemExpress | Get quote | Ask for price |
Description: SB-649701 is a potent human CCR8 antagonist, with a pIC50 of 7.7. AZ084 can be used for the research of asthma[1]. |
SB-269970 |
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HY-15370 | MedChemExpress | 50mg | EUR 854.4 |
Description: SB-269970 is a potent, selective and brain-penetrant 5-HT7 receptor antagonist with a pKi of 8.3. SB-269970 exhibits >50-fold selectivity against other 5-HT receptors[1][2]. |
SB216763 |
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G607 | ABM | 1.0 mg | EUR 225 |
Description: 3-(2,4-dichlorophenyl)-4-(1-methyl-1H-indol-3-yl)-1H-pyrrole-2,5-dione |
SB756050 |
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HY-102016 | MedChemExpress | 50mg | EUR 194.81 |
Description: SB756050 is a selective TGR5 agonist. SB756050 has the potential for type 2 diabetes treatment. |
SB-699551 |
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HY-103100 | MedChemExpress | Get quote | Ask for price |
Description: SB-699551 is a potent and selective 5-HT5A antagonist with a pKi of 8.3[1]. SB-699551 inhibits tumorsphere formation. SB-699551 reduces phosphorylation of AKT at serine residue 473 (S473), WNK1, PRAS40. SB-699551 shows anticancer activity and has the potential for the research of breast tumor[2][3]. |
SB-200646 |
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HY-103129A | MedChemExpress | Get quote | Ask for price |
Description: SB-200646 is the first selective 5-HT2B/2C over 5-HT2A receptor antagonist with pKi values of 7.5, 6.9 and 5.2 for 5-HT2B, 5-HT2C and 5-HT2A, respectively. SB-200646 is orally active and has electrophysiological and anxiolytic properties in vivo[1][2]. |
SB228357 |
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HY-103154 | MedChemExpress | 5mg | EUR 703.47 |
Description: SB228357 is a selective, potent and orall active 5-HT2C/2B receptor antagonist with pKi values of 6.9, 8.0 and 9.0 for 5-HT2A, 5-HT2B and 5-HT2C, respectively. SB228357 has antidepressant/anxiolytic effects[1][2]. |
SB-221284 |
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HY-103155 | MedChemExpress | Get quote | Ask for price |
Description: SB 221284 is a selective 5-HT2C/2B receptor antagonist with pKi values are 6.4, 7.9 and 8.6 for 5-HT2A, 5-HT2B and 5-HT2C receptors, respectively. SB 221284 can be used for the research of neurological disease[1]. |
SB297006 |
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HY-103361 | MedChemExpress | 5mg | EUR 487.02 |
Description: SB297006 is a CCR3 antagonist, which significantly inhibits proliferation and neurosphere formation in CCL11-treated neural progenitor cells. |
SB-328437 |
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HY-103363 | MedChemExpress | 10 mg | EUR 671.01 |
Description: SB-328437 is a potent, selective non-peptide CCR3 antagonist with an IC50 of 4.5 nM[1]. |
SB-205384 |
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HY-103501 | MedChemExpress | 5mg | EUR 660.18 |
Description: SB-205384 is a GABAA receptor modulator. The primary effect of SB-205384 on GABAA-activated currents is a prolonged response decay half-life upon removal of the agonist[1]. |
SB-431542 |
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HY-10431 | MedChemExpress | 100mg | EUR 389.62 |
Description: SB-431542 is a TGF-β receptor kinase inhibitor (TRKI). SB-431542 has inhibitory activity for ALK4, ALK5 and ALK7 with IC50 values of 1 μM, 0.75 μM and 2 μM, respectively. SB-431542 also inhibits TGF-β-induced transcription, gene expression, apoptosis, and growth suppression. SB-431542 can be used for the research of cancer and signal transduction pathways[1][2][3]. |
SB399885 |
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HY-105896 | MedChemExpress | Get quote | Ask for price |
Description: SB399885 is a potent, selective, brain penetrant and orally active 5-HT6 receptor antagonist with pKi values 9.11 and 9.02 for human recombinant and native 5-HT6 receptors, respectively. SB399885 has cognitive enhancing properties[1]. |
SB-705498 |
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HY-10633 | MedChemExpress | 100mg | EUR 773.82 |
Description: SB-705498 is a potent, selective and orally bioavailable transient receptor potential vanilloid 1 (TRPV1) receptor antagonist with a pIC50 of 7.1. |
SB-657510 |
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HY-10656 | MedChemExpress | 10mg | EUR 1298.72 |
Description: SB-657510 is a selective urotensin II (UII) receptor (UT) antagonist. The Ki values are 61, 17, 30, 65 and 56 nM for human, monkey, cat, rat and mouse receptors, respectively. SB-657510 exerts anti-inflammatory effects by inhibiting UII-induced upregulation of inflammatory mediators such as adhesion molecules, cytokines, and tissue factor in human vascular endothelial cells[1][2]. |
SB-611812 |
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HY-10664 | MedChemExpress | 1 mg | EUR 1136.38 |
Description: SB-611812 is a urotensin II receptor (UTR) antagonist with the potential in the research of cardiovascular disease[1][2]. |
SB-218078 |
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HY-107407 | MedChemExpress | 1 mg | EUR 149.35 |
Description: SB-218078 is a potent, selective, ATP-competitive and cell-permeable checkpoint kinase 1 (Chk1) inhibitor that inhibits Chk1 phosphorylation of cdc25C with an IC50 of 15 nM. SB-218078 is less potently inhibits Cdc2 (IC50 of 250 nM) and PKC (IC50 of 1000 nM). SB-218078 causes apoptosis by DNA damage and cell cycle arrest[1][2][3]. |
SB-649868 |
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HY-10806 | MedChemExpress | 100mg | EUR 2532.51 |
Description: SB-649868 is a potent and selective orally active orexin (OX) 1 and OX2 receptor antagonist (pKi =9.4 and 9.5 at the OX1 and OX2 receptor, respectively). |
SB-633825 |
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HY-108333 | MedChemExpress | 10 mg | EUR 2056.31 |
Description: SB-633825 is a potent and ATP-competitive inhibitor of TIE2, LOK (STK10) and BRK with IC50s of 3.5 nM, 66 nM, 150 nM, respectively. SB-633825 can inhibit cancer cell growth and angiogenesis[1]. |
SB-277011 |
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HY-10847 | MedChemExpress | 50mg | EUR 1315.2 |
SB-366791 |
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HY-12245 | MedChemExpress | 10mg | EUR 343.08 |
Description: SB-366791 is a potent and selective vanilloid receptor (VR1/TRPV1) antagonist (IC50=5.7 nM). SB-366791 can be used for the research of inflammation[1][2]. |
SB269652 |
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HY-12324 | MedChemExpress | 100mg | EUR 627.72 |
SB297006 |
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MBS132856-INQUIRE | MyBiosource | INQUIRE | Ask for price |
SB-681323 |
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MBS133317-INQUIRE | MyBiosource | INQUIRE | Ask for price |