PPACK Dihydrochloride

PPACK Dihydrochloride

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H89 Dihydrochloride
20-abx076747
  • EUR 811.20
  • EUR 360.00
  • 25 mg
  • 5 mg

MPP dihydrochloride
B6910-10 10 mg
EUR 381.6

MPP dihydrochloride
B6910-50 50 mg
EUR 1413.6

SAG dihydrochloride
GL1175-1MG 1 mg
EUR 234

SAG dihydrochloride
GL1175-5MG 5 mg
EUR 688.8

TMB (dihydrochloride)
HY-15930A 10mM/1mL
EUR 135.6

SAG dihydrochloride
GL1175-1 1
EUR 98.4

SAG dihydrochloride
GL1175-25 25
EUR 334.3

SAG dihydrochloride
GL1175-5 5
EUR 169

TMB dihydrochloride
TB0514 1g
EUR 85.06

IT1t dihydrochloride
B5650-10 10 mg
EUR 385.2
Description: IT1t dihydrochloride is a potent antagonist of CXCR4 with IC50 value of 8.0 nM [1]. C-X-C chemokine receptor type 4 (CXCR4) is an ?-chemokine receptor for chemokine CXCL12.

IT1t dihydrochloride
B5650-100 100 mg
EUR 2100
Description: IT1t dihydrochloride is a potent antagonist of CXCR4 with IC50 value of 8.0 nM [1]. C-X-C chemokine receptor type 4 (CXCR4) is an ?-chemokine receptor for chemokine CXCL12.

IT1t dihydrochloride
B5650-25 25 mg
EUR 710.4
Description: IT1t dihydrochloride is a potent antagonist of CXCR4 with IC50 value of 8.0 nM [1]. C-X-C chemokine receptor type 4 (CXCR4) is an ?-chemokine receptor for chemokine CXCL12.

IT1t dihydrochloride
B5650-5 5 mg
EUR 243.6
Description: IT1t dihydrochloride is a potent antagonist of CXCR4 with IC50 value of 8.0 nM [1]. C-X-C chemokine receptor type 4 (CXCR4) is an ?-chemokine receptor for chemokine CXCL12.

IT1t dihydrochloride
B5650-5.1 10 mM (in 1mL DMSO)
EUR 261.6
Description: IT1t dihydrochloride is a potent antagonist of CXCR4 with IC50 value of 8.0 nM [1]. C-X-C chemokine receptor type 4 (CXCR4) is an ?-chemokine receptor for chemokine CXCL12.

IT1t dihydrochloride
B5650-50 50 mg
EUR 1232.4
Description: IT1t dihydrochloride is a potent antagonist of CXCR4 with IC50 value of 8.0 nM [1]. C-X-C chemokine receptor type 4 (CXCR4) is an ?-chemokine receptor for chemokine CXCL12.

1400W dihydrochloride
2055-25 each
EUR 405.6

1400W dihydrochloride
2055-5 each
EUR 151.2

DMPQ Dihydrochloride
20-abx076714
  • EUR 693.60
  • EUR 326.40
  • 25 mg
  • 5 mg

DMPQ dihydrochloride
B6642-10 10 mg
EUR 223.2

DMPQ dihydrochloride
B6642-5 5 mg
EUR 184.8

GNTI dihydrochloride
B6669-10 10 mg
EUR 459.6

GNTI dihydrochloride
B6669-50 50 mg
EUR 1746

1400W dihydrochloride
B6730-10 10 mg
EUR 170.4
Description: 1400W dihydrochloride is a potent and selective inhibitor of inducible nitric oxide synthase with Kd value of 7 nM [1]. Inducible nitric oxide synthase (iNOS) is an enzyme catalyzing the production of nitric oxide (NO) and is involved in immune response.

1400W dihydrochloride
B6730-100 100 mg
EUR 873.6
Description: 1400W dihydrochloride is a potent and selective inhibitor of inducible nitric oxide synthase with Kd value of 7 nM [1]. Inducible nitric oxide synthase (iNOS) is an enzyme catalyzing the production of nitric oxide (NO) and is involved in immune response.

1400W dihydrochloride
B6730-50 50 mg
EUR 525.6
Description: 1400W dihydrochloride is a potent and selective inhibitor of inducible nitric oxide synthase with Kd value of 7 nM [1]. Inducible nitric oxide synthase (iNOS) is an enzyme catalyzing the production of nitric oxide (NO) and is involved in immune response.

1400W dihydrochloride
GK6799-100MG 100 mg
EUR 661.2

1400W dihydrochloride
GK6799-25MG 25 mg
EUR 274.8

1400W dihydrochloride
GK6799-5MG 5 mg
EUR 136.8

PAβN (dihydrochloride)
HY-101444A 10mM/1mL
EUR 154.8

IT1t (dihydrochloride)
HY-101458A 10mg
EUR 308.4

1400W (Dihydrochloride)
HY-18731 10mM/1mL
EUR 151.2

DAPI (dihydrochloride)
HY-D0814 50mg
EUR 439.2

1400W dihydrochloride
GK6799-100 100
EUR 605.5

1400W dihydrochloride
GK6799-25 25
EUR 228.1

1400W dihydrochloride
GK6799-5 5
EUR 86.5

GGACK Dihydrochloride
1847-5 5 mg
EUR 382.8
Description: A potent and irreversible inhibitor of Urokinase (uPA (IC??<1 µM), Factor VIIa, Factor IXa, Factor Xa, and trypsin.

GGACK Dihydrochloride
A2582-5 5 mg
EUR 282
Description: A potent and irreversible inhibitor of Urokinase (uPA (IC??<1 µM), Factor VIIa, Factor IXa, Factor Xa, and trypsin.

JDTic (dihydrochloride)
HY-10487 50mg
EUR 1501.2

MS023 (dihydrochloride)
HY-19615B 100mg
EUR 1093.2

DG172 (dihydrochloride)
HY-19737A 50mg
EUR 704.4

GBR 12935 dihydrochloride
B4661-10 10 mg
EUR 129.6

GBR 12935 dihydrochloride
B4661-100 100 mg
EUR 296.4

GBR 12935 dihydrochloride
B4661-50 50 mg
EUR 192

ETP 45835 dihydrochloride
B4938-10 10 mg
EUR 428.4

ETP 45835 dihydrochloride
B4938-50 50 mg
EUR 1608

AZ 10606120 dihydrochloride
B5410-10 10 mg
EUR 408
Description: KD: 1.4 nM and 1.9 nM for human and rat P2X7 receptors, respectivleyThe P2X7 receptor has intriguing biophysical properties, activates a diverse range of cellular events and mediates a wide range of functional effects.

AZ 10606120 dihydrochloride
B5410-50 50 mg
EUR 1531.2
Description: KD: 1.4 nM and 1.9 nM for human and rat P2X7 receptors, respectivleyThe P2X7 receptor has intriguing biophysical properties, activates a diverse range of cellular events and mediates a wide range of functional effects.

CP 99994 dihydrochloride
B5422-10 10 mg
EUR 478.8

CP 99994 dihydrochloride
B5422-50 50 mg
EUR 1824

SB 243213 dihydrochloride
B5444-10 10 mg
EUR 486

SB 243213 dihydrochloride
B5444-50 50 mg
EUR 1802.4

JNJ 5207852 dihydrochloride
B5513-10 10 mg
EUR 289.2

JNJ 5207852 dihydrochloride
B5513-5 5 mg
EUR 180

JNJ 5207852 dihydrochloride
B5513-50 50 mg
EUR 1021.2

A 412997 dihydrochloride
B5639-25 25 mg
EUR 642
Description: A 412997 dihydrochloride is a selective agonist of dopamine D4 receptor with Ki values of 7.9 and 12.1 nM for human and rat D4 receptors, respectively [1]. Dopamine D4 receptor is a G protein-coupled receptor and is activated by dopamine.

A 412997 dihydrochloride
B5639-5 5 mg
EUR 212.4
Description: A 412997 dihydrochloride is a selective agonist of dopamine D4 receptor with Ki values of 7.9 and 12.1 nM for human and rat D4 receptors, respectively [1]. Dopamine D4 receptor is a G protein-coupled receptor and is activated by dopamine.

SA 4503 dihydrochloride
B5778-10 10 mg
EUR 297.6

SA 4503 dihydrochloride
B5778-5.1 10 mM (in 1mL DMSO)
EUR 343.2

SA 4503 dihydrochloride
B5778-50 50 mg
EUR 1069.2

BMS 599626 dihydrochloride
B5792-10 10 mg
EUR 642
Description: BMS 599626 dihydrochloride is a potent and selective inhibitor of EGFR and ErbB2 with IC50 values of 22 and 32 nM, respectively [1].

TC 1698 dihydrochloride
B7089-10 10 mg
EUR 408

TC 1698 dihydrochloride
B7089-50 50 mg
EUR 1531.2

JP 1302 dihydrochloride
B7147-10 10 mg
EUR 466.8

JP 1302 dihydrochloride
B7147-50 50 mg
EUR 1771.2

BYK 191023 dihydrochloride
B7210-10 10 mg
EUR 297.6
Description: IC50: 86 nM for iNOSNO synthases are enzymes responsible for the generation of nitric oxide from the amino acid L-arginine. Once expressed the inducible NO synthase (iNOS) is active and produces ?M concentrations of NO over longer periods.

BYK 191023 dihydrochloride
B7210-5 5 mg
EUR 184.8
Description: IC50: 86 nM for iNOSNO synthases are enzymes responsible for the generation of nitric oxide from the amino acid L-arginine. Once expressed the inducible NO synthase (iNOS) is active and produces ?M concentrations of NO over longer periods.

BYK 191023 dihydrochloride
B7210-50 50 mg
EUR 999.6
Description: IC50: 86 nM for iNOSNO synthases are enzymes responsible for the generation of nitric oxide from the amino acid L-arginine. Once expressed the inducible NO synthase (iNOS) is active and produces ?M concentrations of NO over longer periods.

ARL 17477 dihydrochloride
B7363-10 10 mg
EUR 350.4
Description: ARL 17477 dihydrochloride is a selective and potent neuronal nitrogen oxide synthase (nNOS) inhibitor with IC50 values of 1 and 17?M for nNOS and endothelial NOS, respectively [1].

ARL 17477 dihydrochloride
B7363-50 50 mg
EUR 1264.8
Description: ARL 17477 dihydrochloride is a selective and potent neuronal nitrogen oxide synthase (nNOS) inhibitor with IC50 values of 1 and 17?M for nNOS and endothelial NOS, respectively [1].

PD 168568 dihydrochloride
B7420-10 10 mg
EUR 369.6

PD 168568 dihydrochloride
B7420-50 50 mg
EUR 1363.2

A 943931 dihydrochloride
B7495-10 10 mg
EUR 486
Description: A 943931, is an H4R (one of histamine receptor subtypes) antagonist [1] with high affinities to H4Rs of human (Ki = 5 nM), rat (Ki = 4 nM) and mouse (Kb = 6 nM) [2]. H4R is one of 4 known G-protein-coupled receptors of histamine for histamine to mediate its physiological functions [3].

A 943931 dihydrochloride
B7495-50 50 mg
EUR 1802.4
Description: A 943931, is an H4R (one of histamine receptor subtypes) antagonist [1] with high affinities to H4Rs of human (Ki = 5 nM), rat (Ki = 4 nM) and mouse (Kb = 6 nM) [2]. H4R is one of 4 known G-protein-coupled receptors of histamine for histamine to mediate its physiological functions [3].

PG 01037 dihydrochloride
B7524-10 10 mg
EUR 309.6

PG 01037 dihydrochloride
B7524-25 25 mg
EUR 633.6

PG 01037 dihydrochloride
B7524-5 5 mg
EUR 195.6

WAY 207024 dihydrochloride
B7525-10 10 mg
EUR 576
Description: WAY 207024 dihydrochloride is a potent gonadotropin releasing hormone receptor (GnRH-R) antagonist with IC50 values of 12 and 71 nM for human and rat GnRH receptors, respectively [1].

WAY 208466 dihydrochloride
B7531-10 10 mg
EUR 289.2

WAY 208466 dihydrochloride
B7531-25 25 mg
EUR 582

WAY 208466 dihydrochloride
B7531-5 5 mg
EUR 184.8

WAY 267464 dihydrochloride
B7538-10 10 mg
EUR 556.8

JNJ 10181457 dihydrochloride
B7567-10 10 mg
EUR 466.8

JNJ 10181457 dihydrochloride
B7567-50 50 mg
EUR 1771.2

BMS 470539 dihydrochloride
B7577-10 10 mg
EUR 544.8
Description: BMS 470539 dihydrochloride is a potent and selective melanocortin-1 (MC1) receptor agonist with IC50 of 120 nM [1]. The melanocortin-1 receptor (MC-1R) is a G protein-coupled receptor involved in blocking inflammation and augmenting skin pigmentation [1].

BMS 470539 dihydrochloride
B7577-50 50 mg
EUR 2056.8
Description: BMS 470539 dihydrochloride is a potent and selective melanocortin-1 (MC1) receptor agonist with IC50 of 120 nM [1]. The melanocortin-1 receptor (MC-1R) is a G protein-coupled receptor involved in blocking inflammation and augmenting skin pigmentation [1].

PS 1145 dihydrochloride
B7683-25 25 mg
EUR 428.4

PS 1145 dihydrochloride
B7683-5 5 mg
EUR 164.4

A 331440 dihydrochloride
B7698-10 10 mg
EUR 459.6
Description: A-331440 is described here instead of A-331440 dihydrochloride. A-331440 is an antagonist of non-imidazole histamine H3 receptor with an IC50 value of 22.7 nM for human cortex histamine H3 [1].

A 331440 dihydrochloride
B7698-50 50 mg
EUR 1746
Description: A-331440 is described here instead of A-331440 dihydrochloride. A-331440 is an antagonist of non-imidazole histamine H3 receptor with an IC50 value of 22.7 nM for human cortex histamine H3 [1].

R 1485 dihydrochloride
B7723-10 10 mg
EUR 466.8

R 1485 dihydrochloride
B7723-50 50 mg
EUR 1771.2

DBM 1285 dihydrochloride
B7748-10 10 mg
EUR 517.2

DBM 1285 dihydrochloride
B7748-50 50 mg
EUR 1987.2

LDN 209929 dihydrochloride
B7785-10 10 mg
EUR 466.8
Description: Target: haspin kinaseIC50: 55 nMLDN 209929 dihydrochloride is a selective and potent haspin kinase inhibitor with IC50 value of 55 nM [1]. LDN 209929 dihydrochloride displays 180-fold selectivity on haspin kinase over DYRK2 [1].

LDN 209929 dihydrochloride
B7785-50 50 mg
EUR 1771.2
Description: Target: haspin kinaseIC50: 55 nMLDN 209929 dihydrochloride is a selective and potent haspin kinase inhibitor with IC50 value of 55 nM [1]. LDN 209929 dihydrochloride displays 180-fold selectivity on haspin kinase over DYRK2 [1].

GBR 13069 dihydrochloride
B6296-10 10 mg
EUR 321.6

GBR 13069 dihydrochloride
B6296-50 50 mg
EUR 1167.6

SKF 91488 dihydrochloride
B6331-10 10 mg
EUR 265.2

SKF 91488 dihydrochloride
B6331-50 50 mg
EUR 926.4

GBR 12783 dihydrochloride
B6332-10 10 mg
EUR 303.6

GBR 12783 dihydrochloride
B6332-50 50 mg
EUR 1082.4

BD 1063 dihydrochloride
B6489-10 10 mg
EUR 205.2
Description: BD 1063 dihydrochloride is an antagonist of ?-1 receptor with Ki value of 9.15 nM [1].?-receptor is a type of opioid receptor. There are two subtypes of ?-receptor: ?-1 and ?-2.?-1 receptor plays an important role in stimulating dopamine release and modulating the actions of cocaine [2].

BD 1063 dihydrochloride
B6489-5 5 mg
EUR 151.2
Description: BD 1063 dihydrochloride is an antagonist of ?-1 receptor with Ki value of 9.15 nM [1].?-receptor is a type of opioid receptor. There are two subtypes of ?-receptor: ?-1 and ?-2.?-1 receptor plays an important role in stimulating dopamine release and modulating the actions of cocaine [2].

RS 16566 dihydrochloride
B6548-10 10 mg
EUR 408

RS 16566 dihydrochloride
B6548-50 50 mg
EUR 1531.2

CGP 20712 dihydrochloride
B6552-10 10 mg
EUR 459.6
Description: CGP 20712 dihydrochloride is a potent and selective antagonist of ?1-adrenoceptor with IC50 value of 0.7 nM [1]. ?1-adrenoceptor is a G-protein coupled receptor and mediates uncoupling protein-1 (UCP1) gene expression induced by norepinephrine (NE) [2].

CGP 20712 dihydrochloride
B6552-50 50 mg
EUR 1746
Description: CGP 20712 dihydrochloride is a potent and selective antagonist of ?1-adrenoceptor with IC50 value of 0.7 nM [1]. ?1-adrenoceptor is a G-protein coupled receptor and mediates uncoupling protein-1 (UCP1) gene expression induced by norepinephrine (NE) [2].

CP 93129 dihydrochloride
B6558-10 10 mg
EUR 381.6

CP 93129 dihydrochloride
B6558-50 50 mg
EUR 1413.6

GR 55562 dihydrochloride
B6572-10 10 mg
EUR 400.8

GR 55562 dihydrochloride
B6572-50 50 mg
EUR 1491.6

RJR 2429 dihydrochloride
B6666-10 10 mg
EUR 369.6

RJR 2429 dihydrochloride
B6666-50 50 mg
EUR 1363.2

SCH 79797 dihydrochloride
B6801-10 10 mg
EUR 285.6

SCH 79797 dihydrochloride
B6801-5 5 mg
EUR 223.2

SKF 86002 dihydrochloride
B6921-10 10 mg
EUR 439.2

SKF 86002 dihydrochloride
B6921-50 50 mg
EUR 1654.8

GW 583340 dihydrochloride
B6989-10 10 mg
EUR 439.2

GW 583340 dihydrochloride
B6989-50 50 mg
EUR 1654.8

CGH 2466 dihydrochloride
B7027-10 10 mg
EUR 340.8
Description: CGH 2466 dihydrochloride is a combined adenosine receptor antagonist. It is an inhibitor of phosphodiesterase type 4 and p38 mitogen-activated protein kinase. It inhibited the phosphodiesterase 4D (PDE4D) isoenzyme with an IC50 value of 22±5 nM.

CGH 2466 dihydrochloride
B7027-50 50 mg
EUR 1245.6
Description: CGH 2466 dihydrochloride is a combined adenosine receptor antagonist. It is an inhibitor of phosphodiesterase type 4 and p38 mitogen-activated protein kinase. It inhibited the phosphodiesterase 4D (PDE4D) isoenzyme with an IC50 value of 22±5 nM.

AZ 12080282 dihydrochloride
A8657-10 10 mg
EUR 498
Description: AZ 12080282 dihydrochloride is a selective inhibitor of Hh with IC50 value <0.012 ?M [1]. It is also reported that AZ 12080282 also has a selective inhibition to p38? with low nanomolar potency [1].

AZ 12080282 dihydrochloride
A8657-50 50 mg
EUR 1900.8
Description: AZ 12080282 dihydrochloride is a selective inhibitor of Hh with IC50 value <0.012 ?M [1]. It is also reported that AZ 12080282 also has a selective inhibition to p38? with low nanomolar potency [1].

AY 9944 dihydrochloride
A8658-10 10 mg
EUR 289.2
Description: AY 9944 dihydrochloride is a selective inhibitor of ?7-sterol reductase with IC50 value of 13 nM [1].?7-sterol reductase (Dhcr7) is an enzyme and plays an important role in catalyzing the production of cholesterol from 7-Dehydrocholesterol through using NADPH [2, 3].

AY 9944 dihydrochloride
A8658-25 25 mg
EUR 582
Description: AY 9944 dihydrochloride is a selective inhibitor of ?7-sterol reductase with IC50 value of 13 nM [1].?7-sterol reductase (Dhcr7) is an enzyme and plays an important role in catalyzing the production of cholesterol from 7-Dehydrocholesterol through using NADPH [2, 3].

AY 9944 dihydrochloride
A8658-5 5 mg
EUR 184.8
Description: AY 9944 dihydrochloride is a selective inhibitor of ?7-sterol reductase with IC50 value of 13 nM [1].?7-sterol reductase (Dhcr7) is an enzyme and plays an important role in catalyzing the production of cholesterol from 7-Dehydrocholesterol through using NADPH [2, 3].

CP 31398 dihydrochloride
A4476-10 10 mg
EUR 381.6
Description: CP 31398 dihydrochloride is a potent activator of p53 with maximum tolerated dose of 400 ppm [2].Tumor protein p53 (p53) is a crucial protein in multicellular organisms and plays an important role in preventing cancer formation.

CP 31398 dihydrochloride
A4476-50 50 mg
EUR 1413.6
Description: CP 31398 dihydrochloride is a potent activator of p53 with maximum tolerated dose of 400 ppm [2].Tumor protein p53 (p53) is a crucial protein in multicellular organisms and plays an important role in preventing cancer formation.

GBR 12783 (dihydrochloride)
HY-100968 5mg
EUR 267.6

GBR 12935 (dihydrochloride)
HY-12242 10mg
EUR 142.8

RN 1 dihydrochloride
B2080-25 each
EUR 705.6

RN 1 dihydrochloride
B2080-5 each
EUR 222

H-9 dihydrochloride
B5001-25 25 mg
EUR 217.2

H-9 dihydrochloride
B5001-50 50 mg
EUR 339.6

RN 1 dihydrochloride
B5784-10 10 mg
EUR 447.6
Description: RN 1 dihydrochloride is a potent and selective inhibitor of LSD1 with IC50 value of 70 nM [1].

RN 1 dihydrochloride
B5784-50 50 mg
EUR 1695.6
Description: RN 1 dihydrochloride is a potent and selective inhibitor of LSD1 with IC50 value of 70 nM [1].

PB 28 dihydrochloride
B7107-10 10 mg
EUR 340.8

PB 28 dihydrochloride
B7107-50 50 mg
EUR 1245.6

H-7 dihydrochloride
B6342-10 10 mg
EUR 188.4

H-7 dihydrochloride
B6342-25 25 mg
EUR 360

H-7 dihydrochloride
B6342-5 5 mg
EUR 134.4

H-7 dihydrochloride
B6342-50 50 mg
EUR 584.4

MM 77 dihydrochloride
B6511-10 10 mg
EUR 340.8

MM 77 dihydrochloride
B6511-50 50 mg
EUR 1245.6

H-7 dihydrochloride
9543-25 each
EUR 652.8

H-7 dihydrochloride
9543-5 each
EUR 210

H-8 dihydrochloride
GK6037-10MG 10 mg
EUR 136.8

H-8 dihydrochloride
GK6037-50MG 50 mg
EUR 302.4

H-8 dihydrochloride
GK6037-10 10
EUR 86.5

H-8 dihydrochloride
GK6037-50 50
EUR 210.3

ABT 702 dihydrochloride
B5298-10 10 mg
EUR 494.4
Description: IC50: 1.7 nM for adenosine kinaseAdenosine (ADO) is an endogenous homeostatic inhibitory neuromodulator that reduces cellular excitability at sites of tissue injury and inflammation.

ABT 702 dihydrochloride
B5298-100 100 mg
EUR 2049.6
Description: IC50: 1.7 nM for adenosine kinaseAdenosine (ADO) is an endogenous homeostatic inhibitory neuromodulator that reduces cellular excitability at sites of tissue injury and inflammation.

ABT 702 dihydrochloride
B5298-5 5 mg
EUR 331.2
Description: IC50: 1.7 nM for adenosine kinaseAdenosine (ADO) is an endogenous homeostatic inhibitory neuromodulator that reduces cellular excitability at sites of tissue injury and inflammation.

ABT 702 dihydrochloride
B5298-5.1 10 mM (in 1mL DMSO)
EUR 379.2
Description: IC50: 1.7 nM for adenosine kinaseAdenosine (ADO) is an endogenous homeostatic inhibitory neuromodulator that reduces cellular excitability at sites of tissue injury and inflammation.

ABT 702 dihydrochloride
B5298-50 50 mg
EUR 1417.2
Description: IC50: 1.7 nM for adenosine kinaseAdenosine (ADO) is an endogenous homeostatic inhibitory neuromodulator that reduces cellular excitability at sites of tissue injury and inflammation.

C 021 dihydrochloride
B5457-1 1 mg
EUR 135.6
Description: C 021 dihydrochloride is a potent antagonist of CCR4 with IC50 values of 0.039 and 0.14 ?M for inhibition of chemotaxis in mouse and human, respectively [1].

C 021 dihydrochloride
B5457-5 5 mg
EUR 309.6
Description: C 021 dihydrochloride is a potent antagonist of CCR4 with IC50 values of 0.039 and 0.14 ?M for inhibition of chemotaxis in mouse and human, respectively [1].

TCN 237 dihydrochloride
B5523-10 10 mg
EUR 320.4

TCN 237 dihydrochloride
B5523-5 5 mg
EUR 254.4

VU 590 dihydrochloride
B7526-10 10 mg
EUR 284.4

VU 590 dihydrochloride
B7526-50 50 mg
EUR 1004.4

ML 786 dihydrochloride
B7736-10 10 mg
EUR 583.2
Description: IC50: 2.1, 2.5 and 4.2 nM for B-RafV600E, C-Raf and wild-type B-Raf, respectivelyML 786 is a potent Raf kinase inhibitor.

ARC 239 dihydrochloride
B6508-25 25 mg
EUR 642
Description: ARC 239 dihydrochloride is a selective antagonist of ?2B adrenoceptor with pKD value of 8.8 [1]. ?2B adrenoceptor is a G-protein coupled receptor.

ARC 239 dihydrochloride
B6508-5 5 mg
EUR 212.4
Description: ARC 239 dihydrochloride is a selective antagonist of ?2B adrenoceptor with pKD value of 8.8 [1]. ?2B adrenoceptor is a G-protein coupled receptor.

XE 991 dihydrochloride
B6917-10 10 mg
EUR 214.8

XE 991 dihydrochloride
B6917-5 5 mg
EUR 141.6

XE 991 dihydrochloride
B6917-50 50 mg
EUR 714

AMN 082 dihydrochloride
B7034-10 10 mg
EUR 284.4
Description: AMN 082 dihydrochloride is an specific allosteric agonist of mGluR7 [1]. In the absence of orthosteric agonist, AMN 082 activated the human mGlu7 receptor with an EC50 of 64 nM in vitro [2].

AMN 082 dihydrochloride
B7034-50 50 mg
EUR 1004.4
Description: AMN 082 dihydrochloride is an specific allosteric agonist of mGluR7 [1]. In the absence of orthosteric agonist, AMN 082 activated the human mGlu7 receptor with an EC50 of 64 nM in vitro [2].

SA4503 dihydrochloride
B3046-25 25 mg
EUR 612

SA4503 dihydrochloride
B3046-5 5 mg
EUR 199.2

AT7867 dihydrochloride
A3199-10 10 mg
EUR 408
Description: IC50: AKT1 32 nM, AKT2 17 nM, AKT3 47 nM, PKA 20 nMThe serine/threonine kinase AKT plays a pivotal role in signal transduction events involved in malignant transformation and chemoresistance and is an attractive target for the development of cancer therapeutics.

AT7867 dihydrochloride
A3199-100 100 mg
EUR 2210.4
Description: IC50: AKT1 32 nM, AKT2 17 nM, AKT3 47 nM, PKA 20 nMThe serine/threonine kinase AKT plays a pivotal role in signal transduction events involved in malignant transformation and chemoresistance and is an attractive target for the development of cancer therapeutics.

AT7867 dihydrochloride
A3199-5 5 mg
EUR 320.4
Description: IC50: AKT1 32 nM, AKT2 17 nM, AKT3 47 nM, PKA 20 nMThe serine/threonine kinase AKT plays a pivotal role in signal transduction events involved in malignant transformation and chemoresistance and is an attractive target for the development of cancer therapeutics.

AT7867 dihydrochloride
A3199-5.1 10 mM (in 1mL DMSO)
EUR 344.4
Description: IC50: AKT1 32 nM, AKT2 17 nM, AKT3 47 nM, PKA 20 nMThe serine/threonine kinase AKT plays a pivotal role in signal transduction events involved in malignant transformation and chemoresistance and is an attractive target for the development of cancer therapeutics.

AT7867 dihydrochloride
A3199-50 50 mg
EUR 1537.2
Description: IC50: AKT1 32 nM, AKT2 17 nM, AKT3 47 nM, PKA 20 nMThe serine/threonine kinase AKT plays a pivotal role in signal transduction events involved in malignant transformation and chemoresistance and is an attractive target for the development of cancer therapeutics.

LDK378 dihydrochloride
A3544-10 10 mg
EUR 186
Description: LDK378 is a highly potent inhibitor of anaplastic lymphoma kinase (ALK), which is a receptor tyrosine kinase belonging to the superfamily of insulin receptor, with half maximal inhibitory concentration IC50 of 200 pM.

LDK378 dihydrochloride
A3544-100 100 mg
EUR 331.2
Description: LDK378 is a highly potent inhibitor of anaplastic lymphoma kinase (ALK), which is a receptor tyrosine kinase belonging to the superfamily of insulin receptor, with half maximal inhibitory concentration IC50 of 200 pM.

PPACK Dihydrochloride